Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 12:11:18 UTC 2023
by
admin
on
Sat Dec 16 12:11:18 UTC 2023
|
| Protein Type | ENZYME |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
4APO0P2BE7
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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4APO0P2BE7
Created by
admin on Sat Dec 16 12:11:19 UTC 2023 , Edited by admin on Sat Dec 16 12:11:19 UTC 2023
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PRIMARY | |||
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O60341
Created by
admin on Sat Dec 16 12:11:19 UTC 2023 , Edited by admin on Sat Dec 16 12:11:19 UTC 2023
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PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IRREVERSIBLE INHIBITOR
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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RADIOLIGAND->TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
PRECLINICAL
IC50
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INHIBITOR -> TARGET |
Binds rapidly and irreversibly to the
FAD cofactor in KDM1A.
IC50
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INHIBITOR -> TARGET |
99.33% INHIBITION @ 0.4 MICROMOLAR
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INHIBITOR -> TARGET |
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![Structure of rel-trans-4-Amino-N-[(1R,2S)-2-phenylcyclopropyl]cyclohexanemethanamine](/img/bf7c4374-47c6-447e-a0ac-eb999265da0e.svg "Structure of rel-trans-4-Amino-N-[(1R,2S)-2-phenylcyclopropyl]cyclohexanemethanamine")
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
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| MOL_WEIGHT | CHEMICAL |
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