OPROZOMIB

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National Institutes of Health Divider Arrow

NCATS

Details

Stereochemistry	ABSOLUTE
Molecular Formula	C25H32N4O7S
Molecular Weight	532.609
Optical Activity	UNSPECIFIED
Defined Stereocenters	4 / 4
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure of OPROZOMIB

Structure Search

SMILES

COC[C@H](NC(=O)[C@H](COC)NC(=O)C1=CN=C(C)S1)C(=O)N[C@@H](CC2=CC=CC=C2)C(=O)[C@@]3(C)CO3

InChI

InChIKey=SWZXEVABPLUDIO-WSZYKNRRSA-N

InChI=1S/C25H32N4O7S/c1-15-26-11-20(37-15)24(33)29-19(13-35-4)23(32)28-18(12-34-3)22(31)27-17(21(30)25(2)14-36-25)10-16-8-6-5-7-9-16/h5-9,11,17-19H,10,12-14H2,1-4H3,(H,27,31)(H,28,32)(H,29,33)/t17-,18-,19-,25+/m0/s1

HIDE SMILES / InChI

Molecular Formula	C25H32N4O7S
Molecular Weight	532.609
Charge	0
Count

Stereochemistry	ABSOLUTE
Additional Stereochemistry	No
Defined Stereocenters	4 / 4
E/Z Centers	0
Optical Activity	UNSPECIFIED

Approval Year

Substance Class	Chemical Created by `admin` on `Sat Dec 16 01:30:38 UTC 2023` Edited by `admin` on `Sat Dec 16 01:30:38 UTC 2023`
Record UNII	MZ37792Y8J
Record Status	`Validated (UNII)`
Record Version

Download

Name

Type

Language

OPROZOMIB

Official Name

English

O-METHYL-N-((2-METHYLTHIAZOL-5-YL)CARBONYL)-L-SERYL-O-METHYL-N-((1S)-1-BENZYL-2-((2R)- 2-METHYLOXIRAN-2-YL)-2-OXOETHYL)-L-SERINAMIDE

Systematic Name

English

ONX-0912

Code

English

oprozomib [INN]

Common Name

English

PR-047

Common Name

English

ONX 0912

Code

English

OPROZOMIB [USAN]

Common Name

English

Oprozomib [WHO-DD]

Common Name

English

Classification Tree Code System Code

FDA ORPHAN DRUG

449614

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

FDA ORPHAN DRUG

443614

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

NCI_THESAURUS

C2160

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

Code System Code Type Description

EVMPD

SUB126055

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

PUBCHEM

25067547

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

FDA UNII

MZ37792Y8J

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

CAS

935888-69-0

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

EPA CompTox

DTXSID201025950

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

USAN

YY-148

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

NCI_THESAURUS

C91388

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

WIKIPEDIA

Oprozomib

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

INN

9597

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

DRUG BANK

DB11991

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

SMS_ID

100000151658

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

ChEMBL

CHEMBL2103884

Created by admin on Sat Dec 16 01:30:38 UTC 2023 , Edited by admin on Sat Dec 16 01:30:38 UTC 2023

PRIMARY

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OPROZOMIB

ACTIVE MOIETY