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Details

Stereochemistry ACHIRAL
Molecular Formula C17H15N5O
Molecular Weight 305.3339
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of ZALEPLON

SMILES

CCN(C(C)=O)C1=CC=CC(=C1)C2=CC=NC3=C(C=NN23)C#N

InChI

InChIKey=HUNXMJYCHXQEGX-UHFFFAOYSA-N
InChI=1S/C17H15N5O/c1-3-21(12(2)23)15-6-4-5-13(9-15)16-7-8-19-17-14(10-18)11-20-22(16)17/h4-9,11H,3H2,1-2H3

HIDE SMILES / InChI
Molecular Formula C17H15N5O
Molecular Weight 305.3339
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Approval Year

Unknown
86413
Substance Class Chemical
Created
by admin
on Fri Dec 15 15:41:39 UTC 2023
Edited
by admin
on Fri Dec 15 15:41:39 UTC 2023
Record UNII
S62U433RMH
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ZALEPLON
EMA EPAR   INN   JAN   MART.   MI   ORANGE BOOK   USAN   VANDF   WHO-DD  
USAN   INN  
Official Name English
ZALEPLON CIV
USP-RS  
Common Name English
ZALEPLON [MART.]
Common Name English
ZAL-846
Code English
ZALEPLON [USP MONOGRAPH]
Common Name English
ACETAMIDE, N-(3-(3-CYANOPYRAZOLO(1,5-.ALPHA.)PYRIMIDIN-7-YL)PHENYL)-N-ETHYL-
Common Name English
ZALEPLON CIV [USP-RS]
Common Name English
LJC10846
Code English
ZALEPLON [USAN]
Common Name English
L-846
Code English
3'-(3-CYANOPYRAZOLO(1,5-.ALPHA.)PYRIMIDIN-7-YL)-N-ETHYLACETANILIDE
Common Name English
ZALEPLON [MI]
Common Name English
CL 284,846
Code English
LJC-10846
Code English
ZERENE
Brand Name English
SKP-1041
Code English
CL-284846
Code English
ZALEPLON [VANDF]
Common Name English
zaleplon [INN]
Common Name English
Zaleplon [WHO-DD]
Common Name English
ZALEPLON [ORANGE BOOK]
Common Name English
SONATA
Brand Name English
L846
Code English
ZALEPLON [JAN]
Common Name English
ZALEPLON [EMA EPAR]
Common Name English
Classification Tree Code System Code
EMA ASSESSMENT REPORTS SONATA (AUTHORIZED: SLEEP INITIATION AND MAINTENANCE DISORDERS)
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
EMA ASSESSMENT REPORTS ZERENE (WITHDRAWN: SLEEP INITIATION AND MAINTENANCE DISORDERS)
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
NDF-RT N0000183360
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
NCI_THESAURUS C29756
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
DEA NO. 2781
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
WHO-VATC QN05CF03
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
LIVERTOX NBK548924
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
WHO-ATC N05CF03
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
Code System Code Type Description
NCI_THESAURUS
C29551
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
LACTMED
Zaleplon
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
FDA UNII
S62U433RMH
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
SMS_ID
100000088001
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
CAS
151319-34-5
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
WIKIPEDIA
ZALEPLON
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
CHEBI
10102
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
RXCUI
74667
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY RxNorm
MESH
C085665
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
ChEMBL
CHEMBL1521
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
IUPHAR
4345
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
DRUG BANK
DB00962
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
RS_ITEM_NUM
1724350
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
DRUG CENTRAL
2857
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
USAN
GG-36
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
DAILYMED
S62U433RMH
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
EVMPD
SUB00132MIG
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
EPA CompTox
DTXSID5023748
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
PUBCHEM
5719
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
MERCK INDEX
m11579
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY Merck Index
INN
7312
Created by admin on Fri Dec 15 15:41:39 UTC 2023 , Edited by admin on Fri Dec 15 15:41:39 UTC 2023
PRIMARY
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GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1
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Structure of ZALEPLON
BASIS OF STRENGTH->SUBSTANCE
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Process impurity; may not be found in all manufacturing processes
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Structure of ISOZALEPLON
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Structure of N-(3-(3-(DIMETHYLAMINO)ACRYLOYL)PHENYL)-N-ETHYLACETAMIDE, (E)-
IMPURITY -> PARENT
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Structure of N-DESESETHYLZALEPLON
IMPURITY -> PARENT
Process impurity; may not be found in all manufacturing processes
CHROMATOGRAPHIC PURITY (HPLC/UV)
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Structure of 7-(3-(N-ETHYLACETAMIDO)PHENYL)PYRAZOLO(1,5-A)PYRIMIDINE-3-CARBOXAMIDE
IMPURITY -> PARENT
Process impurity; may not be found in all manufacturing processes.
CHROMATOGRAPHIC PURITY (HPLC/UV)
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Related Record Type Details
Structure of ZALEPLON
ACTIVE MOIETY
Name Property Type Amount Referenced Substance Defining Parameters References
Volume of Distribution PHARMACOKINETIC
Biological Half-life PHARMACOKINETIC
NIH
NCATS
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