U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 09:09:02 UTC 2023
Edited
by admin
on Sat Dec 16 09:09:02 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
SMV73KW49C
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ENSEREPTIDE
INN  
INN  
Official Name English
PXL01
Code English
PXL-01
Code English
ACETYL(HUMAN LACTOTRANSFERRIN-(15-39)-PEPTIDAMIDE)
Common Name English
ensereptide [INN]
Common Name English
Code System Code Type Description
NCI_THESAURUS
C169952
Created by admin on Sat Dec 16 09:09:02 UTC 2023 , Edited by admin on Sat Dec 16 09:09:02 UTC 2023
PRIMARY
FDA UNII
SMV73KW49C
Created by admin on Sat Dec 16 09:09:02 UTC 2023 , Edited by admin on Sat Dec 16 09:09:02 UTC 2023
PRIMARY
PUBCHEM
49863418
Created by admin on Sat Dec 16 09:09:02 UTC 2023 , Edited by admin on Sat Dec 16 09:09:02 UTC 2023
PRIMARY
CAS
254433-51-7
Created by admin on Sat Dec 16 09:09:02 UTC 2023 , Edited by admin on Sat Dec 16 09:09:02 UTC 2023
PRIMARY
INN
9579
Created by admin on Sat Dec 16 09:09:02 UTC 2023 , Edited by admin on Sat Dec 16 09:09:02 UTC 2023
PRIMARY
From To
1_5 1_22
Related Record Type Details
TARGET->INHIBITOR OF EXPRESSION
TARGET->INHIBITOR OF EXPRESSION
TARGET->ACTIVATOR OF EXPRESSION
Increased expression of PRG4 mRNA in tendons treated with rabPXL01 in HA, but not in tendon sheaths. In addition, treatment with rabPXL01 in HA led to repression of the mRNA levels for the pro-inflammatory mediators interleukin (IL)-1β, IL-6, and IL-8 in tendon sheaths.
TARGET->INHIBITOR OF EXPRESSION
Increased expression of PRG4 mRNA in tendons treated with rabPXL01 in HA, but not in tendon sheaths. In addition, treatment with rabPXL01 in HA led to repression of the mRNA levels for the pro-inflammatory mediators interleukin (IL)-1β, IL-6, and IL-8 in tendon sheaths.
Related Record Type Details
ACTIVE MOIETY
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL